Browsing by Author Dreassi, Elena
Showing results 1 to 8 of 8
Issue Date | Title | Author(s) |
---|---|---|
2022 | Antibacterial alkylguanidino ureas: Molecular simplification approach, searching for membrane-based MoA | D'Agostino, Ilaria; Ardino, Claudia; Poli, Giulio; Sannio, Filomena; Lucidi, Massimiliano; Poggialini, Federica; Visaggio, Daniela; Rango, Enrico; Filippi, Silvia; Petricci, Elena; Visca, Paolo; Lorenzo Botta ; Docquier, Jean-Denis; Dreassi, Elena |
2023 | Biological Evaluation and In Vitro Characterization of ADME Profile of In-House Pyrazolo[3,4-d]pyrimidines as Dual Tyrosine Kinase Inhibitors Active against Glioblastoma Multiforme | Poggialini, Federica; Vagaggini, Chiara; Brai, Annalaura; Pasqualini, Claudia; Crespan, Emmanuele; Maga, Giovanni; Perini, Cecilia; Cabella, Noemi; Botta, Lorenzo ; Musumeci, Francesca; Frosini, Maria; Schenone, Silvia; Dreassi, Elena |
2016 | Development and in Vitro Evaluation of a Microbicide Gel Formulation for a Novel Non-Nucleoside Reverse Transcriptase Inhibitor Belonging to the N-Dihydroalkyloxybenzyloxopyrimidines (N-DABOs) Family | Tintori, Cristina; Brai, Annalaura; Dasso Lang, Maria Chiara; Deodato, Davide; Greco, Antonia Michela; Bizzarri, Bruno Mattia ; Cascone, Lorena; Casian, Alexandru; Zamperini, Claudio; Dreassi, Elena; Crespan, Emmanuele; Maga, Giovanni; Vanham, Guido; Ceresola, Elisa; Canducci, Filippo; Ariƫn, Kevin K; Botta, Maurizio |
2023 | Discovery and Optimization of a Novel Macrocyclic Amidinourea Series Active as Acidic Mammalian Chitinase Inhibitors | Balestri, Lorenzo Jacopo Ilic; Trivisani, Claudia Immacolata; Orofino, Francesco; Fiorucci, Diego; Truglio, Giuseppina Ivana; D'Agostino, Ilaria; Poggialini, Federica; Botta, Lorenzo ; Docquier, Jean-Denis; Dreassi, Elena |
2022 | Focused library of phenyl-fused macrocyclic amidinoureas as antifungal agents | Balestri, Lorenzo J I; D'Agostino, Ilaria; Rango, Enrico; Vagaggini, Chiara; Marchitiello, Rosalba; Mariotti, Melinda; Casian, Alexandru; Deodato, Davide; Truglio, Giuseppina I; Orofino, Francesco; Sanguinetti, Maurizio; Bugli, Francesca; Lorenzo Botta ; Dreassi, Elena |
2022 | Privileged Scaffold Decoration for the Identification of the First Trisubstituted Triazine with Anti-SARS-CoV-2 Activity | Cesarini, Silvia; Vicenti, Ilaria; Poggialini, Federica; Secchi, Massimiliano; Giammarino, Federica; Varasi, Ilenia; Lodola, Camilla; Zazzi, Maurizio; Dreassi, Elena; Maga, Giovanni; Botta, Lorenzo ; Saladino, Raffaele |
2022 | The impact of counterions in biological activity: case study of antibacterial alkylguanidino ureas | Ardino, Claudia; Sannio, Filomena; Pasero, Carolina; Botta, Lorenzo ; Dreassi, Elena; Docquier, Jean-Denis; D'Agostino, Ilaria |
2023 | Tyrosine Kinase Inhibitor Si409 Has In Vitro and In Vivo Anti-Tumor Activity Against Diffuse Large B-Cell Lymphoma | Rango, Enrico; Di Maria, Salvatore; Zamperini, Claudio; Poggialini, Federica; Crespan, Emmanuele; Perini, Cecilia; Sabetta, Samantha; Saponara, Simona; Fusi, Fabio; Maga, Giovanni; Angelucci, Adriano; Gaudio, Eugenio; Berton, Francesco; Schenone, Silvia; Botta, Lorenzo ; Dreassi, Elena; Botta, Maurizio |